Clavulanic acid

Clavulanic acid yog ib yam khoom tshwj xeeb uas sib koom tes nrog penicillinases thiab ua rau lawv tsis zoo. Nws tuaj yeem pom nyob rau hauv cov lus sau ntawm feem ntau ua ke muaj zog tshuaj. Ntxiv nrog, clavulanic acid tuaj yeem siv rau hauv cov lus qhia nrog beta-lactam antibiotics.

Lub mechanism ntawm kev txiav txim ntawm clavulanic acid

Kws txawj ntse clavulanic acid rau cov metabolism. Cov tshuaj yeeb dej cawv no muaj peev xwm ua tau cov tshuaj tua kabmob antimicrobial. Cov tshuaj uas muaj clavulanic acid yog siv los siv rau ntau yam kab mob uas tshwm sim los ntawm kab mob thiab kab mob.

Cov qauv ntawm molecules ntawm clavulanic acid yog zoo li cov tshuaj tiv thaiv ntawm penicillin series. Tias yog vim li cas lawv cov kev sib xyaw los ntawm lub chaw tshuaj ntsuam pom tau pom zoo tshwj xeeb. Lub ntsiab qhov txawv yog tias hauv cov kua qaub es tsis thiazolidine muaj ib lub nplhaib oxazolidine. Tab sis qhov kev sib tw ntawm cov tshuaj yog tsis muaj kev cuam tshuam dab tsi.

Mus rau hauv lub cev, clavulanic acid inhibits beta-lactamase - bacterial enzymes, cov tsos ntawm uas contributes rau qhov tseem ceeb ua si ntawm teeb meem microorganisms. Feem ntau, txoj cai ntawm kev txiav txim ntawm clavulanic acid yog yooj yim: los ntawm kev tiv thaiv lub plhaub, nws nkag mus rau hauv lub hlwb cov kab mob thiab "tua" cov enzymes nyob hauv. Yog li, cov khoom tsis tso cai rau cov kab mob thiab cov kab mob ua rau kom muab.

Raws li kev xyaum tau pom, tom qab qhov kev tua, qhov txo ntawm beta-lactamase yog suav hais tias yuav luag tsis tau. Vim yog cov kab mob pathogenic no tsis tuaj yeem tsim muaj, tab sis kuj plam lub sijhawm los tiv thaiv cov tshuaj tua kab mob uas ua rau lawv tsis ua haujlwm.

Cov kev ua tau zoo ntawm cov khoom muaj qis heev. Txawm tias cov kab mob ntawm cov kab mob thiab cov kab mob uas tau tswj kom muaj kev tiv thaiv tawm tsam Amoxicillin thiab Ampicillin raug rhuav tshem los ntawm qhov kev txiav txim ntawm clavulanic acid. Ntawd yog, qhov tshwm sim ntawm kev siv tshuaj ua ke yog ntau dua li ntawm cov tshuaj tua kab mob.

Yeej, cov tshuaj siv nrog cov tshuaj clavulinic acid yog noj qhov ncauj, tab sis qee kis, lawv cov kev tso dej tshuaj tso cai yog qhov zoo tshaj. Yog li, tsis muaj qhov tsis haum rau kev khwv noj khwv haus, nws tsis haum rau cov neeg mob uas muaj kev tsis txaus siab. Hauv cov rooj plaub tshwj xeeb, clavulic acid nrog Amoxicillin thiab Ticarcillin tuaj yeem raug txawm los ntawm cov poj niam cev xeeb tub.

Augmentin - Amoxicillin nrog clavulanic acid

Qhov no yog ib qho ntawm cov tshuaj tua kab mob zoo tshaj plaws. Cov tshuaj yog muaj nrog cov kev kuaj mob xws li:

Qov ntawm Augmentin rau txhua tus neeg mob tau xaiv ib tus zuj zus, nyob ntawm daim ntawv thiab qhov tsis yooj yim ntawm tus kab mob, qhov mob ntawm tus neeg mob, nws lub hnub nyoog, sib tw kuaj mob. Kev kho nrog cov tshuaj yuav tsum tsis pub tsawg dua tsib zaug, tab sis tsis pub ntau tshaj kaum plaub hnub.

Flemoxin nrog clavulanic acid

Qhov no yog lwm txoj kev paub zoo, hu ua Flemoklav. Tus kab mob tua tau tus kab mob zoo me ntsis ntau tshaj qhov tseem ceeb tshaj plaws ntawm cov tshuaj Flemoxin, tab sis nws tus nqi yog kev lees paub los ntawm nws txoj kev ua haujlwm zoo.

Ib lub cuab tam siv los kho ntau yam kev mob hlab:

Flemoklav yog tso tawm rau hauv daim ntawv ntawm cov ntsiav tshuaj soluble, vim tias nws cov hauj lwm tseem ceeb ntau dua.