Nimesil thiab cawv

Cov tshuaj tiv thaiv ua kom tsis muaj zog tiv thaiv qee zaum kuj muaj tshuaj tua kab mob hauv lub cev. Tus neeg sawv cev raws li kev txiav txim tsis siv rau lawv, txawm tias nws yog ib qhov kev xav zoo heev. Cuaj kaum, Nimesil thiab cawv categorically tsis tau noj nyob rau hauv ib hnub, vim hais tias qhov no yuav ua rau irreversible teebmeem nyob rau hauv lub cev.

Nimesil thiab cawv sib luag

Cleavage ntawm ethyl cawv tshwm sim nyob rau hauv daim siab, thaum ua ib yam tshuaj lom hu ua acetaldehyde. Feem ntau ntawm cov dej cawv tsis ua rau mob cancer tuag, qhov uas haus dej cawv yog ua rau hloov cov ntaub so ntswg los ntawm cov ntaub so ntswg. Yog li, muaj dej muaj zog muaj cov nyhuv tshuaj lom ntawm lub cev, rhuav tshem cov kab mob siab. Lub cev tivthaiv ntawm Nimesil yog qhov khoom ua si, ib qho tshuaj tsis-steroidal anti-inflammatory substance, ntxiv rau anesthetizing, ua rau ib tug antipyretic nyhuv. Nws yog ib qho qaug zog toxin, uas, zoo li acetaldehyde, muaj peev xwm ua kom puas siab puas hlwb cov tshuaj tom qab txhaj tshuaj ntau tshaj li cov tau pom zoo hauv cov lus qhia. Hauv cov kev mob tshwm sim rau cov yeeb tshuaj, nws tau qhia tias ib qho kev tsis zoo ntawm kev kho tshuaj yuav yog qhov txhaum cai ntawm lub siab ua haujlwm, thiab kev sib kis kab mob siab . Yog li no, Nimesil thiab cawv yog tsis tsim nyog los ua ke, vim tib lub sijhawm siv cov tshuaj phem rau lub koom haum nrhiav ntshav ua ke txhawb lawv txoj haujlwm.

Puas yog nws ua tau noj Namsil cawv, thiab lawv txoj kev sib raug zoo yog dabtsi?

Nyob rau hauv kev qhia rau cov tshuaj piav qhia, tsis muaj ib qho kev qhia tias Nimesil thiab cawv tsis ua raws, thiab tsis piav qhia txog cov mechanisms ntawm kev sib raug zoo. Tab sis nws yuav tsum tau sau tseg tias cov metabolizers (cleavage) ntawm nimesulide tshwm sim nrog kev koom tes ntawm ib qho tshwj xeeb enzyme - isoenzyme cytochrome. Raws li nws muab tawm, nws kuj txhawb nqa qhov kev ua txhaum ntawm ethanol tebchaw hauv daim siab. Yog li, lub simultaneous siv cov tshuaj nrog cawv provokes ntev li ntawm no enzyme thiab, raws li ib tug consequence, ib qho kev nce nyob rau hauv qhov mob load on daim siab.

Ntxiv mus, vim yog tsis muaj kev tshawb fawb ntawm Nimesil cov kev sib tshuam nrog muaj zog haus, tsis muaj pov thawj ntawm qhov ua tau zoo npaum li cas qhov cuab yeej no yuav ua kom loog. Ntawm cov kws txawj, nws ntseeg tau hais tias cawv blocks kev ua ntawm yeeb tshuaj, thiab kev txiav txim txaus ntawm qhov analgesic tsis tiav.

Ib qho ntawm feem ntau yuav raug kev phem ntawm kev noj haus Namsim nrog cawv yog lub sijhawm tsis tuaj yeem ntes cov teebmeem ntawm kev khomob xws li sab hauv lub plab hauv cov hlwv hauv plab vim kev qaug. Hauv lub xeev tsis nco qab lawm, tsis quav ntsej txog qhov teeb meem no yuav ua rau tuag taus.

Nimesil tom qab dej cawv - raug mob

Muaj qee zaum muaj thaum tom qab noj mov yog muaj mob taub hau heev los yog mob tsis zoo, nrog rau kev hnov ​​mob tsis xis nyob. Lawm, koj xav tau sai sai tshem tawm tsis xis nyob thiab feem ntau siv Nimesil rau qhov no. Nws yog ib qho tseem ceeb kom nco ntsoov tias qhov sib txawv nruab nrab ntawm qhov kawg ntawm cov dej cawv, txawm tias tsis muaj zog, piv txwv li, npias, thiab noj cov tshuaj yuav tsum tsawg kawg yog 6 teev. Thaum lub sij hawm no, feem ntau ntawm cov cawv cawv yuav tsum metabolized nyob rau hauv daim siab thiab tshem tawm ntawm lub bile thiab los ntawm ob lub raum. Txawm hais tias qhov muaj txiaj ntsim zoo ntawm cov tshuaj acetaldehyde tseem yuav ua rau siab, nws tsis tuaj yeem mob siab rau qhov zoo li cov nyhuv ntawm nimesulide, thiab qhov kev kho mob ntawm tus mob hnyav yuav nyob ruaj ntseg. Txawm li cas los xij, nws raug pom zoo kom hloov cov tshuaj no nrog ib tus neeg tsis muaj tshuaj lom (Aspirin, Ibuprom) kom tsis txhob muaj qhov tsis zoo rau lub siab.